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CRTh2 antagonist 3

Cat. No.: IBDI-436730

CRTh2 antagonist 3 is a potent chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTh2) antagonist. CRTh2 antagonist 3 enhances the activity of PDK1 toward a short peptide substrate, with an EC50 of 2 μM and a Kd of 8.4 μM. CRTh2 antagonist 3 has the potential for cardiovascular inflammation.

Size (Solid):

Product Details

Target Prostaglandin Receptor | PDK-1
Molecular Weight 356.44
SMILES O=C(O)CN1C2=CC=CC=C2N=C1SCCOC3=C(C)C=CC=C3C

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.