GSK2798745

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Cat. No.: IBDI-434267

GSK2798745 is a potent, selective, and orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively. GSK2798745 can be used in cardiac and respiratory diseases research.

Size (Solution): 10 mM * 1 mL in DMSO

Size (Solid + Solvent): 10 mM * 1 mL ready for reconstitution

Size (Solid):

Product Details

Target	TRP Channel
Molecular Weight	460.53
Appearance	Solid
SMILES	N#CC1=CC=C2N=CN(C[[email protected]](CCC3)(C)C[[email protected]@]43CN(C5=NC=C(C(C)(O)C)N=C5)C(O4)=O)C2=C1
Purity	99.46%

Storage & Handling

Shipping	Room temperature in continental US. May vary elsewhere.
Storage	Powder: -20°C/3 years; 4°C/2 years In solvent: -80°C/6 months; -20°C/1 month
Regulatory Status	This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.

! For research use only, not intended for any clinical use.