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KDM2A/7A-IN-1

Cat. No.: IBDI-432687

KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16 μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive on methyl transferases, and histone acetyl transferases.

Size (Solid):

Product Details

Target Histone Demethylase
Molecular Weight 506.68
Appearance Solid
SMILES CC(N([[email protected]@H](C1=CN=CC(CCCCCCCN2CCCC2)=C1)[[email protected]@]3(C4=CC=CC=C4)C#N)C5=C3C=CC=C5)=O
Purity 99.57%

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Powder: -20°C/3 years; 4°C/2 years
In solvent: -80°C/6 months; -20°C/1 month
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.