Mu opioid receptor antagonist 1

Cat. No.: IBDI-434754

Mu opioid receptor antagonist 1 (compound 19) is a selective and orally active μ opioid receptor (MOR) ligand with an Ki value of 0.58 nM and an EC50 of 1.15 nM. Orally administrating with Mu opioid receptor antagonist 1 increases intestinal motility during morphine-induced constipation. Mu opioid receptor antagonist 1 can be used for researching opioid-induced constipation (OIC).

Product Details

Target	Opioid Receptor
Molecular Weight	436.50
SMILES	O[[email protected]]12[[email protected]]3CC4=C5[[email protected]@]1(CCN3CC6CC6)[[email protected]]([[email protected]@H](CC2)NC(C7=CN=CN7)=O)OC5=C(O)C=C4

Storage & Handling

Shipping	Room temperature in continental US. May vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status	This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.