OARV-771

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Cat. No.: IBDI-432882

OARV-771 is a VHL-based BET degrader (PROTAC) with improved cell permeability. OARV-771 shows DC50s of 6, 1, and 4 nM for Brd4, Brd2 and Brd3, respectively.

Size (Solution): 10 mM * 1 mL in DMSO

Size (Solid + Solvent): 10 mM * 1 mL ready for reconstitution

Size (Solid):

Product Details

Target	Epigenetic Reader Domain \| PROTACs
Molecular Weight	987.62
Appearance	Solid
SMILES	CC1=C(C)SC2=C1C(C3=CC=C(C=C3)Cl)=N[[email protected]@H](CC(OCCOCCCOCC(N[[email protected]@H](C(C)(C)C)C(N4[[email protected]@H](C[[email protected]](C4)O)C(N[[email protected]](C5=CC=C(C6=C(C)N=CS6)C=C5)C)=O)=O)=O)=O)C7=NN=C(C)N27
Purity	98.33%

Storage & Handling

Shipping	Room temperature in continental US. May vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status	This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.

! For research use only, not intended for any clinical use.