P300 bromodomain-IN-1

Cat. No.: IBDI-433873

P300 bromodomain-IN-1 (Compoun 1u) is a potent p300 (EP300) bromodomain inhibitor with an IC50 of 49 nM. P300 bromodomain-IN-1 suppresses the expression of c-Myc and induces G1/G0 phase arrest and apoptosis in OPM-2 cells.

Product Details

Target	Epigenetic Reader Domain | Histone AcetyltransfeRase
Molecular Weight	535.03
SMILES	COC1=CC=C(C=C1Cl)N2C(C[[email protected]]2C3=NC4=CC(C5=C(ON=C5C)C)=CC=C4N3[[email protected]]6CC[[email protected]@H](CC6)OC)=O

Storage & Handling

Shipping	Room temperature in continental US. May vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status	This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.