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* Please note that all of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.

PERK-IN-5

Cat. No.: IBDI-433086

PERK-IN-5 is a highly potent, selectively and orally bioavailable PERK inhibitor (IC50s of 2 and 9 nM for PERK and p-eIF2α, respectively). PERK-IN-5 can significantly inhibit tumor growth in the 786-O renal cell carcinoma xenograft tumor model.

Size (Solid):

Product Details

Target PERK
Molecular Weight 468.50
Appearance Solid
SMILES CCC1=C(C2=CN=C(N)C(C(NC(C)C)=O)=C2)C=CC(NC([[email protected]@H](C3=CC(F)=CC(F)=C3)O)=O)=C1
Purity 99.40%

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Powder: -20°C/3 years; 4°C/2 years
In solvent: -80°C/6 months; -20°C/1 month
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.
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