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PU139

Cat. No.: IBDI-437288

PU139 is a potent pan-histone acetyltransferase (HAT) inhibitor. PU139 blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB (cAMP response element-binding) protein (CBP) and p300 with IC50s of 8.39, 9.74, 2.49 and 5.35 μM, respectively.

Size (Solid):

Product Details

Target Histone AcetyltransfeRase
Molecular Weight 246.26
Appearance Solid
SMILES O=C1N(C2=CC=C(F)C=C2)SC3=NC=CC=C31
Purity 98.03%

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.