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(R)-GSK-3685032

Cat. No.: IBDI-434205

(R)-GSK-3685032 is the R-enantiomer of GSK-3685032. GSK-3685032 is a non-time-dependent, noncovalently, first-in-class reversible DNMT1-selective inhibitor, with an IC50 of 0.036 μM. GSK-3685032 induces robust loss of DNA methylation, transcriptional activation, and cancer cell growth inhibition.

Size (Solid):

Product Details

Target DNA MethyltransfeRase
Molecular Weight 420.53
Appearance Solid
SMILES N#CC1=C(N2CCC(CC2)N)N=C(C(C#N)=C1CC)S[[email protected]](C3=CC=CC=C3)C(N)=O
Purity 98.02%

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.
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