RP101075

Cat. No.: IBDI-434235

RP101075, an active metabolite of Ozanimod, is a potent, orally active S1PR (sphingosine-1-phosphate receptor 1) agonist, with an EC50 of 0.27 nM. RP101075 displays >100-fold selectivity over S1PR5 (EC50=5.9 nM) and >10000-fold over S1PR 2, 3, and 4. RP101075 displays superior cardiovascular safety profile.

Product Details

Target	LPL Receptor | Drug Metabolite
Molecular Weight	360.41
SMILES	N#CC1=CC(C2=NC(C3=CC=CC4=C3CC[[email protected]@H]4N)=NO2)=CC=C1OC(C)C

Storage & Handling

Shipping	Room temperature in continental US. May vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status	This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.