S1427

Cat. No.: IBDI-436075

S1427 is a tranylcypromine-derived LSD1 inhibitor with the IC50 of 390 nM and Ki of 80 nM. S1427 exhibits desirable hERG channel inhibition and microsomal stability profiles. Inhibition of LSD1 partially reduces the proliferation of cancer cells.

Product Details

Target	Histone Demethylase
Molecular Weight	474.52
SMILES	O=C(N1CCC2(CC1)CCNC2)CN[[email protected]]3C[[email protected]@H]3C4=C(C(F)=CC(F)=C4)OCC5=CC=CN=C5F

Storage & Handling

Shipping	Room temperature in continental US. May vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status	This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.