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* Please note that all of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.

SSR240612

Cat. No.: IBDI-437748

SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist, with Kis of 0.48 nM and 0.73 nM for B1 kinin receptors of human fibroblast MRC5 and HEK cells expressing human B1 receptors, 481 nM and 358 nM for B2 receptors of guinea pig ileum membranes and CHO cells expressing human B1 receptor, respectively.

Size (Solid):

Product Details

Target Bradykinin Receptor
Molecular Weight 793.41
Appearance Solid
SMILES O=S(N[[email protected]@H](C1=CC=C2C(OCO2)=C1)CC(N[[email protected]@H](C(N(C)C(C)C)=O)CC3=CC=C(CN([[email protected]@H]4C)[[email protected]](CCC4)C)C=C3)=O)(C5=CC(C=CC(OC)=C6)=C6C=C5)=O.Cl[H]
Purity 99.51%

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.
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