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SY-5609

Cat. No.: IBDI-434220

SY-5609 (CDK7-IN-3) is an orally active, highly selective, noncovalent CDK7 inhibitor with a KD of 0.065 nM. SY-5609 shows poor inhibition on CDK2 (Ki=2600 nM), CDK9 (Ki=960 nM), CDK12 (Ki=870 nM). SY-5609 induces apoptosis in tumor cells and has antitumor activity.

Size (Solid):

Product Details

Target CDK | Apoptosis
Molecular Weight 490.46
Appearance Solid
Synonyms CDK7-IN-3
SMILES N#CC1=C(P(C)(C)=O)C2=C(C=C1)C(C3=NC(N[[email protected]@H]4CNC(C)(C)CC4)=NC=C3C(F)(F)F)=CN2
Purity 99.66%

Storage & Handling

Shipping Room temperature in continental US. May vary elsewhere.
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Regulatory Status This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use.
! For research use only, not intended for any clinical use.
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