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Amelparib

Cat. No: CDIA-1354

CAS. No.: 1227156-72-0

Synonyms: JPI-289

Size: 50 mg

Price: Inquiry

Product Details
Formula	C19H25N3O3
Molecular Weight	343.42
Smiles String	O=C1C2=C(C3=C(C=C(C=C3N1)CN4CCOCC4)OCC)NCCC2

Storage & Handling
Shipping	Room temperature.
Storage	Please refer to the instruction manual.

Description

Amelparib is a potent, orally active, and water-soluble inhibitor of PARP-1. Amelparib inhibits PARP-1 activity (IC50 =18.5 nmol/L) and cellular PAR formation (IC50 =10.7 nmol/L) in the nanomolar range. Amelparib is a potential neuroprotective agent. Amelparib has the potential for the research of acute ischaemic stroke.

! For research use only. Not intended for any clinical use.