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Aprocitentan-d4

Cat. No: CDIA-2022

Synonyms: ACT-132577 d4

Size: 10 mg

Price: Inquiry

Product Details
Formula	C16H10D4Br2N6O4S
Molecular Weight	550.22
Appearance	Solid
Purity	97.39%
Smiles String	O=S(N)(NC1=NC=NC(OC([2H])([2H])C([2H])([2H])OC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)=O

Storage & Handling
Shipping	Room temperature.
Storage Powder	-20 °C/3 years, 4 °C/2 years

Description

Aprocitentan-d4 is a deuterium labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively.

! For research use only. Not intended for any clinical use.