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Aprocitentan

Cat. No: CDIA-1004

CAS. No.: 1103522-45-7

Synonyms: ACT-132577

Size: 5 mg

Price: Inquiry

Product Details
Formula	C16H14Br2N6O4S
Molecular Weight	546.19
Appearance	Solid
Purity	98.13%
Smiles String	O=S(N)(NC1=NC=NC(OCCOC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)=O

Storage & Handling
Shipping	Room temperature.
Storage Powder	-20 °C/3 years, 4 °C/2 years

Description

Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively.

! For research use only. Not intended for any clinical use.