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Azepexole di hydrochloride

Cat. No: CDIA-1693

CAS. No.: 36067-72-8

Synonyms: B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride

Size: 50 mg

Price: Inquiry

Product Details
Formula	C9H17Cl2N3O
Molecular Weight	254.16
Smiles String	NC(O1)=NC2=C1CCN(CC)CC2.[H]Cl.[H]Cl

Storage & Handling
Shipping	Room temperature.
Storage	Please refer to the instruction manual.

Description

Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM).

! For research use only. Not intended for any clinical use.