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GRK5-IN-4

Cat. No: CDIA-1954

CAS. No.: 2410794-89-5

Synonyms: CCG-265328

Size: 50 mg

Price: Inquiry

Product Details
Formula	C26H25N7O3
Molecular Weight	483.52
Smiles String	O=C(NCC1=CC=C(C(OC)=C1)NC2=NC(NC3=C(C(NC)=O)C=CC=C3)=C4C=CNC4=N2)C#CC

Storage & Handling
Shipping	Room temperature.
Storage	Please refer to the instruction manual.

Description

GRK5-IN-4 (Compound 16d, CCG-265328) is a potent and and selective covalent GRK5 (G protein-coupled receptor kinase 5) inhibitor, with an IC50 of 1.1 μM. GRK5-IN-4 shows 90-fold selectivity over GRK2. GRK5-IN-4 can be used for heart failure research.

! For research use only. Not intended for any clinical use.