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MRS2395

Cat. No: CDIA-1889

CAS. No.: 491611-55-3

Size: 50 mg

Price: Inquiry

Product Details
Formula	C20H30ClN5O4
Molecular Weight	439.94
Smiles String	CNC1=C2N=CN(CC(COC(C(C)(C)C)=O)COC(C(C)(C)C)=O)C2=NC(Cl)=N1

Storage & Handling
Shipping	Room temperature.
Storage	Please refer to the instruction manual.

Description

MRS2395, an dipivaloyl derivative, is a potent P2Y12 receptor antagonist. MRS2395 inhibits ADP-induced platelet activation with a Ki of 3.6 μM. MRS2395 inhibits cAMP induced by ADP in rat platelets in the presence of PGE1 with an IC50 of 7 µM. MRS2395 enhances platelet dense granule release in response to TRAP-6.

! For research use only. Not intended for any clinical use.