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Nepicastat

Cat. No: CDIA-1276

CAS. No.: 173997-05-2

Synonyms: SYN117; RS-25560-197

Size: 50 mg

Price: Inquiry

Product Details
Formula	C14H15F2N3S
Molecular Weight	295.35
Smiles String	FC1=CC(F)=C2CC[[email protected]@H](CC2=C1)N3C(CN)=CNC3=S

Storage & Handling
Shipping	Room temperature.
Storage	Please refer to the instruction manual.

Description

Nepicastat (SYN117) is a selective, potent, and orally active inhibitor of dopamine-beta-hydroxylase. Nepicastat (SYN117) produces concentration-dependent inhibition of bovine (IC50=8.5 nM) and human (IC50=9 nM) dopamine-beta-hydroxylase. Nepicastat (SYN117) can cross the blood-brain barrier (BBB).

! For research use only. Not intended for any clinical use.