Cat.#: ASSD-138
Description | A3AR covalent antagonist.Binds irreversibly. Apparent pKi values at A3ARs are 6.9 and 8.0 (after 4h), where a Ki shift indicates a covalent mode of action. |
Size | 50 μg |
Chemical Name | 4-[3-(8-Methoxy-2,4-dioxo-3-propylpurino[7,8-a]pyridin-1-yl)propylcarbamoyl]benzenesulfonyl fluoride |
Molecule Weight | 517.5 |
Molecular formula | C23H24FN5O6S |
PubChem identifier | 155513958 |
Purity | >95% |
Solubility | Soluble in DMSO |
Storage | Store at -20° C |
Shipping | Shipped at 4°C |
Cat.# | Name | Size | Price |
---|---|---|---|
ASSD-227 | Organo/Limonene Mount (AC227) | 100 ml | inquiry |
ASSD-192 | 4-Fluoro-7-nitrobenzofurazan (AC192) | 5 mg, 25 mg, 50 mg | inquiry |
ASSD-153 | Brilliant Blue G (AC153) | 1g | inquiry |
ASSD-155 | Bromophenol blue (AC155) | 5g | inquiry |
ASSD-107 | Modified Mayer's Hematoxylin (AC107) | 125 mL, 250 mL, 2×250mL | inquiry |
ASSD-228 | ImmunoHistoMount (AC228) | 30 ml | inquiry |
ASSD-110 | Picro Sirius Red Stain Kit (AC110) | 1 kit, 100 tests | inquiry |
ASSD-215 | 1-Pyrenylmethyl Methanethiosulfonate (AC215) | 10 mg | inquiry |
ASSD-117 | Annexin V-PE Apoptosis Staining / Detection Kit (AC117) | 1 kit, 100 tests | inquiry |
ASSD-223 | Antifade Fluorescence Mounting Medium (aqueous) (AC223) | 10 mL | inquiry |