Cat.#: ASSD-137
| Description | Chemokine CCR2 covalent negative allosteric modulator (NAM) binds intracellularly and forms a covalent bond with one of three proximal cysteine residues of CCR2. Apparent pKi values at CCR2 are 8.7 and 9.2 (after 4h), where a Ki shift indicates a covalent mode of action. |
| Size | 50 μg |
| Chemical Name | 2-[[4-[4-Chloro-2-[[4-chloro-3-(trifluoromethyl)phenyl]sulfonylamino]phenoxy]benzoyl]amino]ethyl thiocyanate |
| Molecule Weight | 590.4 |
| Molecular formula | C23H16Cl2F3N3O4S2 |
| PubChem identifier | 162666730 |
| Purity | >95% |
| Solubility | Soluble in DMSO |
| Storage | Store at -20° C |
| Shipping | Shipped at 4°C |
| Cat.# | Name | Size | Price |
|---|---|---|---|
| ASSD-214 | 8-Aminopyrene-1,3,6-trisulfonic acid trisodium salt (AC214) | 10 mg | inquiry |
| ASSD-215 | 1-Pyrenylmethyl Methanethiosulfonate (AC215) | 10 mg | inquiry |
| ASSD-213 | Fluorescein 6-Maleimide (AC213) | 25 mg, 250 mg | inquiry |
| ASSD-191 | Fluorescein 6-Isothiocyanate, Isomer 2, 95% (AC191) | 100 mg | inquiry |
| ASSD-216 | K 114 (AC216) | 10 mg, 50 mg | inquiry |
| ASSD-186 | Bromocresol Purple (AC186) | 5 g, 10 g | inquiry |
| ASSD-115 | 7-Amino-4-methylcoumarin (AC115) | 100 mg, 500 mg, 1 g | inquiry |
| ASSD-228 | ImmunoHistoMount (AC228) | 30 ml | inquiry |
| ASSD-138 | A3AR covalent antagonist (AC138) | 50 μg | inquiry |
| ASSD-102 | DAPI (AC102) | 10 mg, 50 mg | inquiry |
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