Cat.#: ASSD-139
| Description | Adenosine A1AR Affinity-Based Probe (AfBP) incubate with live cells or membrane fractions can selectively label the desired receptor in the presence of other proteins. AfBP acts as a partial agonist which is highly specific to the A1AR and binds covalently. Apparent pKi values at A1AR are 7.8 and 9.5 (following a 4h preincubation), where a Ki shift indicates a covalent mode of action. |
| Size | 50 μg |
| Applications | For use in confocal microscopy, SDS-PAGE and chemical proteomics profiling applications. |
| Chemical Name | 4-((3-((6-Amino-4-(benzo[d][1,3]dioxol-5-yl)-3,5-dicyanopyridin-2-yl)thio)propyl)(prop-2-yn-1-yl)carbamoyl)benzenesulfonyl fluoride |
| Molecule Weight | 577.6 |
| Molecular formula | C27H20FN5O5S2 |
| PubChem identifier | 167312224 |
| Purity | >95% |
| Solubility | Soluble in DMSO |
| Storage | Store at -20° C |
| Shipping | Shipped at 4°C |
| Cat.# | Name | Size | Price |
|---|---|---|---|
| ASSD-125 | Fluorescent D1 antagonist [SKF83566-green] (AC125) | 50 μg | inquiry |
| ASSD-137 | CCR2 covalent NAM (AC137) | 50 μg | inquiry |
| ASSD-167 | Fura-2 AM (Cell permeant) (AC167) | 1 mg | inquiry |
| ASSD-198 | NHS-5(6)Carboxyrhodamine (AC198) | 25 mg | inquiry |
| ASSD-119 | Fluorescent adenosine agonist [NECA] (AC119) | 500 μg | inquiry |
| ASSD-171 | Ionomycin calcium salt (AC171) | 1mg, 5mg | inquiry |
| ASSD-143 | Fluorescently labeled Muscimol TMR-X conjugate (AC143) | 1mg | inquiry |
| ASSD-220 | Nitrofluorescein, Isomer 2 (AC220) | 1 g | inquiry |
| ASSD-147 | Rhodamine phalloidin-TRITC (AC147) | 300 tests, 100μg | inquiry |
| ASSD-179 | 8-Azidoadenosine-5′-diphosphate Sodium Salt (AC179) | 1 mg, 5 mg | inquiry |
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