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Pizotifen malate

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Specification

Cat. No.

SMD1109

Related Diseases

Depression

Product Name

Pizotifen malate

Size

100.0mg; 200.0mg; 500.0mg; 1.0g; 2.0g; 5.0g

Price

Inquiry

Availability

2 Weeks

Description

Pizotifen, also known as Pizotyline, is a benzocycloheptene-based drug used as a medicine, primarily as a preventative to reduce the frequency of recurrent migraine headaches. Pizotifen is a serotonin antagonist acting mainly at the 5-HT2A and 5HT2C receptors. It also has some activity as an antihistamine as well as some anticholinergic activity.

CAS Number

5189-11-7 (malate)

Chemical Formula

C23H27NO5S

Molecular Weight

429.531

Elemental Analysis

C, 64.32; H, 6.34; N, 3.26; O, 18.62; S, 7.46

Synonym

Pizotyline malate; BC-105 malate; Litec malate; Pizotifen malate; Sanomtgran.

IUPAC/Chemical Name

4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thiophen-4-ylidene)-1-methylpiperidine malate

InChi Key

IWAWCPZVTXCFKD-UHFFFAOYSA-N

InChi Code

InChI=1S/C19H21NS.C4H6O5/c1-20-11-8-15(9-12-20)19-16-5-3-2-4-14(16)6-7-18-17(19)10-13-21-18;5-2(4(8)9)1-3(6)7/h2-5,10,13H,6-9,11-12H2,1H3;2,5H,1H2,(H,6,7)(H,8,9)

SMILES Code

CN1CC/C(CC1)=C2C3=CC=CC=C3CCC4=C\2C=CS4.OC(CC(O)=O)C(O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.