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TAK-653

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Specification

Cat. No.

SMD1195

Related Diseases

Depression

Product Name

TAK-653

Size

5.0mg

Price

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Availability

2 Weeks

Description

TAK-653 is a novel AMPA receptor potentiator, strictly potentiating a glutamate-induced Ca2+ influx in hGluA1i-expressing CHO cells through structural interference at Ser743 in GluA1,

CAS Number

1358751-06-0

Chemical Formula

C19H23N3O3S

Exact Mass

373.146

Molecular Weight

373.471

Elemental Analysis

C, 61.10; H, 6.21; N, 11.25; O, 12.85; S, 8.58

Synonym

TAK-653; TAK653; TAK 653; NBI-1065845; NBI1065845; NBI 1065845; osavampator

IUPAC/Chemical Name

9-(4-(cyclohexyloxy)phenyl)-7-methyl-3,4-dihydropyrazino[2,1-c][1,2,4]thiadiazine 2,2-dioxide

InChi Key

PXJBHEHFVQVDDS-UHFFFAOYSA-N

InChi Code

InChI=1S/C19H23N3O3S/c1-14-13-22-11-12-26(23,24)21-19(22)18(20-14)15-7-9-17(10-8-15)25-16-5-3-2-4-6-16/h7-10,13,16H,2-6,11-12H2,1H3

SMILES Code

CC1=CN(CC2)C(C(C3=CC=C(OC4CCCCC4)C=C3)=N1)=NS2(=O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.