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Tampramine fumarate

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Specification

Cat. No.

SMD1207

Related Diseases

Depression

Product Name

Tampramine fumarate

Size

Customizable

Price

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Description

Tampramine (AHR-9,377) is a tricyclic antidepressant (TCA) which was developed in the 1980s but was never marketed. Despite being a TCA, it acts as a selective norepinephrine reuptake inhibitor and has negligible affinity for adrenergic, histaminergic, and muscarinic receptors.

CAS Number

83166-18-1

Chemical Formula

C27H28N4O4

Exact Mass

472.2111

Molecular Weight

472.55

Elemental Analysis

C, 68.63; H, 5.97; N, 11.86; O, 13.54

Synonym

Tampramine fumarate; AHR 9377; AHR-9377; AHR9377

IUPAC/Chemical Name

11H-Pyrido(2,3-b)(1,4)benzodiazepine-11-propanamine, N,N-dimethyl-6-phenyl-, (E)-2-butenedioate (1:1)

InChi Key

USQAILMOWHOBTK-WLHGVMLRSA-N

InChi Code

InChI=1S/C23H24N4.C4H4O4/c1-26(2)16-9-17-27-21-14-7-6-12-19(21)22(18-10-4-3-5-11-18)25-20-13-8-15-24-23(20)27;5-3(6)1-2-4(7)8/h3-8,10-15H,9,16-17H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1+

SMILES Code

CN(C)CCCN1C2=NC=CC=C2N=C(C3=CC=CC=C3)C4=CC=CC=C41.O=C(O)/C=C/C(O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4℃ for short term (days to weeks), or -20℃ for long term (months).

HS Tariff Code

2934.99.9001

All of our services and products are intended for preclinical research use only and cannot be used to diagnose, treat or manage patients.